ORGNWednesday, August 19, 2009

8:10 AM-12:00 PM Walter E. Washington Convention Center -- Ballroom B, Oral
Technical Achievements in Organic Chemistry Award Symposium
Organizer:Molly E. Hoke
8:10 AMIntroductory Remarks
8:15 AM7-Substituted benzoxazepinones: Novel non-eroidal progesterone receptor modulators
Jeffrey C. Kern, Thomas J. Berrodin, Jeff Cohen, Andrew Fensome, Cheryl Mugford, Eugene A. Terefenko, Ray J. Unwalla, Richard C. Winneker, Matthew R. Yudt, Puwen Zhang, Zhiming Zhang, Yuan Zhu, Jay Wrobel
8:45 AMOvercoming low exposure due to hydrolysis and oxidative metabolism
Cornelia J Forster
9:15 AMPreparation and reactions of pyranoindazole cyclic carbonates
Pete Delgado
9:45 AMSynthesis of LY459477, a conformationally restricted glutamic acid analog
David W. Hoard, Eric D. Moher, Bret A. Astleford, John L. Bowers, Joseph H. Kennedy, Tianwei Ma, Steven M. Massey, John M. McGill III, James A. Monn, Joseph L. Phillips, Michael L. Phillips, Andrew M. Ratz, David K. Robbins, V. Scott Sharp, Roger W. Tharp-Taylor, Allie E. Tripp, Joseph T. Turpin, Matthew J. Valli, Eldon E. Van Meter, Jeffery A. Ward, James M. Dunigan, Jennifer M. Tinsley
10:15 AMIntermission
10:25 AMStructure-based design, synthesis and biological evaluation of novel dihydropyrones as potent HCV RNA polymerase inhibitors
Maria Angelica Linton, Hui Li, John H. Tatlock, Javier Gonzalez, Tanya Jewell, Leena Patel
10:55 AMBenzimidazole based inhibitors of the Gonadotropin releasing hormone
Daniel Green, Jeffrey Pelletier, Murty V. Chengalvala, Joshua E. Cottom, Irene Feingold, Diane Hauze, Christine Huselton, Gregory S. Kopf, Joseph Lundquist, John Mehlmann, John Rogers, Linda Shanno, Jay Wrobel
11:25 AMSynthesis and development of potent Chk1 kinase inhibitors
Shaei Huang, Rob Garbaccio, Edward S. Tasber, Mark E. Fraley, Justin T. Steen, Youwei Yan, Sanjieev Munshi, Mari Ikuta, Lawrence Kuo, Constantine Kreatsoulas, Michael Reilly, Elizabeth Mahan, Steve Stirdivant, Bob Drakas, Keith Rickert, Eileen Walsh, Kelly Hamilton, Carolyn A. Buser, James Hardwick, Xianzhi Mao, Steve Beck, Marc Abrams, Weikang Tao, Rob Lobell, Laura Sepp-Lorenzino, George D. Hartman
11:55 AMConcluding Remarks

Technical Achievements in Organic Chemistry Award Symposium -- Next Session

Symposium Grid -- Division of Organic Chemistry -- Session Listing

The 238th ACS National Meeting, Washington, DC, August 16-20, 2009