| ORGN | Wednesday, August 19, 2009 | ||
8:10 AM-12:00 PM Walter E. Washington Convention Center -- Ballroom B, Oral | |||
Technical Achievements in Organic Chemistry Award Symposium | |||
| Sponsored by: | ORGN | ||
| Organizer: | Molly E. Hoke | ||
| 8:10 AM | Introductory Remarks | ||
| 8:15 AM | 528 | 7-Substituted benzoxazepinones: Novel non-eroidal progesterone receptor modulators Jeffrey C. Kern, Thomas J. Berrodin, Jeff Cohen, Andrew Fensome, Cheryl Mugford, Eugene A. Terefenko, Ray J. Unwalla, Richard C. Winneker, Matthew R. Yudt, Puwen Zhang, Zhiming Zhang, Yuan Zhu, Jay Wrobel | |
| 8:45 AM | 529 | Overcoming low exposure due to hydrolysis and oxidative metabolism Cornelia J Forster | |
| 9:15 AM | 530 | Preparation and reactions of pyranoindazole cyclic carbonates Pete Delgado | |
| 9:45 AM | 531 | Synthesis of LY459477, a conformationally restricted glutamic acid analog David W. Hoard, Eric D. Moher, Bret A. Astleford, John L. Bowers, Joseph H. Kennedy, Tianwei Ma, Steven M. Massey, John M. McGill III, James A. Monn, Joseph L. Phillips, Michael L. Phillips, Andrew M. Ratz, David K. Robbins, V. Scott Sharp, Roger W. Tharp-Taylor, Allie E. Tripp, Joseph T. Turpin, Matthew J. Valli, Eldon E. Van Meter, Jeffery A. Ward, James M. Dunigan, Jennifer M. Tinsley | |
| 10:15 AM | Intermission | ||
| 10:25 AM | 532 | Structure-based design, synthesis and biological evaluation of novel dihydropyrones as potent HCV RNA polymerase inhibitors Maria Angelica Linton, Hui Li, John H. Tatlock, Javier Gonzalez, Tanya Jewell, Leena Patel | |
| 10:55 AM | 533 | Benzimidazole based inhibitors of the Gonadotropin releasing hormone Daniel Green, Jeffrey Pelletier, Murty V. Chengalvala, Joshua E. Cottom, Irene Feingold, Diane Hauze, Christine Huselton, Gregory S. Kopf, Joseph Lundquist, John Mehlmann, John Rogers, Linda Shanno, Jay Wrobel | |
| 11:25 AM | 534 | Synthesis and development of potent Chk1 kinase inhibitors Shaei Huang, Rob Garbaccio, Edward S. Tasber, Mark E. Fraley, Justin T. Steen, Youwei Yan, Sanjieev Munshi, Mari Ikuta, Lawrence Kuo, Constantine Kreatsoulas, Michael Reilly, Elizabeth Mahan, Steve Stirdivant, Bob Drakas, Keith Rickert, Eileen Walsh, Kelly Hamilton, Carolyn A. Buser, James Hardwick, Xianzhi Mao, Steve Beck, Marc Abrams, Weikang Tao, Rob Lobell, Laura Sepp-Lorenzino, George D. Hartman | |
| 11:55 AM | Concluding Remarks | ||
Technical Achievements in Organic Chemistry Award Symposium -- Next Session
Symposium Grid -- Division of Organic Chemistry -- Session Listing
The 238th ACS National Meeting, Washington, DC, August 16-20, 2009