Engineering protein stability using polyethylene glycol conjugation: GCSF as a case study

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Rahul S. Rajan, rrajan@amgen.com1, Tiansheng Li, tli@amgen.com1, Christopher Sloey1, Mohini Aras, m_aras@uclink.berkeley.edu2, Weston Sutherland1, and David N. Brems3. (1) Department of Pharmaceutics, Amgen, Inc, One Amgen Center Drive 2-1-A, Thousand Oaks, CA 91320, (2) University of California at Berkeley, Berkeley, CA 94720, (3) Pharmaceutics Department, Amgen Inc, One Amgen Center Dr, Thousand Oaks, CA 91320
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Protein Sci. 2006 May;15(5):1063-75.