MEDISunday, March 25, 2007

9:00 AM-1:00 PM McCormick Place Lakeside -- Room E353 A/B, Level 3, Oral
Fragment-Based Drug Discovery
Organizer, Presiding:Jeffrey S. Albert
9:00 AMFragment based drug design
Michael Shapiro
9:40 AMFragment screening and its application to drug design: The discovery of low molecular weight, non-peptidic, nanomolar inhibitors of beta-secretase
Philip D Edwards
10:20 AMFragment to lead evolution using chemical microarray screening
Hans-Dieter Junker, Thomas Neumann, Inge Ott, Klaus Burkert, Oliver Keil, Kristina Schmidt, Renate Sekul
11:00 AMStructure activity relationships by mass spectrometry: Discovery of novel MMP3 inhibitors
Denise A. Ockey, Tom R. Gadek
11:40 AMFragment-based drug discovery: From crystal to clinic
Steven Howard
12:20 PMStrategies and experiences in fragment-based drug discovery
Roderick E Hubbard

Symposium Grid -- Division of Medicinal Chemistry -- Session Listing

Symposium Grid -- Biotechnology -- Session Listing

The 233rd ACS National Meeting, Chicago, IL, March 25-29, 2007