| MEDI | Tuesday, 12 September 2006 | ||
1:30 PM-5:00 PM Moscone Center -- Room 102, Oral | |||
Gamma and Beta Secretase | |||
| Sponsored by Biotage | |||
| Organizers: | Andrew W. Stamford Wenge Zhong | ||
| 1:30 PM | Introductory Remarks | ||
| 1:35 PM | 286 | Secretases as therapeutic targets in Alzheimer's disease Martin Citron | |
| 2:05 PM | 287 | Cyclic sulfonamides as γ-secretase inhibitors for the treatment of Alzheimer's disease Dmitri Pissarnitski, Zhiqiang Zhao, Theodros Asberom, Thomas Bara, John W. Clader, William J. Greenlee, Henry Guzik, Lynn Hyde, Hubert Josien, Wei Li, Eric M. Parker, Murali Rajagopalan, Lili Zhang, Amin Nomeir | |
| 2:40 PM | 288 | Design and synthesis of potent gamma secretase inhibitors for the disease-modifying treatment of Alzheimer's Disease Boyd L. Harrison, Anthony Kreft, Asaf Alimardanov, Madeline Antane, Suzan Aschmies, Kevin Atchison, David Casebier, Michael Chlenov, Derek C. Cole, Thomas Comery, George Diamantidis, John W. Ellingboe, Kristi Fan, Cathleen Gonzalez, Diane B. Hauze, Yun Hu, Donna Huryn, Uday Jain, Mei Jin, Dennis Kubrak, Kristina Kutterer, Melissa Lin, Peimin Lu, Joseph Lundquist, Charles Mann, Robert Martone, Scott C. Mayer, William J. Moore, Aram Oganesian, Alex Porte, Lynn Resnick, David Riddell, June Sonnenberg-Reines, Joseph R. Stock, Shaiu-Ching Sun, Eric Wagner, Zhang Wang, Kevin Woller, Zheng Xu, Margaret Zaleska, Minsheng Zhang, Hua Zhou, J. Steven Jacobsen | |
| 3:15 PM | 289 | Structure-based design of potent and highly selective memapsin 2 (BACE) inhibitors Arun K. Ghosh | |
| 3:50 PM | 290 | Design of an efficacious class of BACE inhibitors Hsiu-Chiung Yang, Javier Agejas, David M Bender, Howard Broughton, Ana Belen Bueno, Robert Dally, Timothy Durham, Jon A. Erickson, Juan Espinosa, Rosario Gonzalaz, Patric Hahn, Debra Laigle, Todd Kohn, Patrick C. May, Juan Ramon Rodriguez, Gema Sanz, Timothy A. Shepherd, David Timm, Paloma Vidal, James R. McCarthy | |
| 4:25 PM | 291 | Discovery of 2,6-isonicotinamide beta-secretase inhibitors bearing a primary amine as an aspartate ligand Shaun R. Stauffer | |
Symposium Grid -- Division of Medicinal Chemistry -- Session Listing
Symposium Grid -- Drug Discovery -- Session Listing
The 232nd ACS National Meeting, San Francisco, CA, September 10-14, 2006