TOXITuesday, 12 September 2006

2:00 PM-5:15 PM Moscone Center -- Room 308, Oral
Drug Toxicity & Safety Prediction
Organizers:F. P. Guengerich
Nicholas A. Meanwell
2:00 PMStrategies to reduce drug candidate failure due to off-target activities
Bruce D. Car
2:45 PMStructural basis of drug binding to hERG K+ channels
Michael C Sanguinetti
3:30 PMIntermission
3:45 PMProperties of the hERG potassium channel that promote promiscuous binding of small organic molecules
Robert Pearlstein, Ramy Farid, Tyler Day, Richard Friesner
4:30 PMThe hERG channel: Tuned in? Chemical strategies for dialing out an off-target source of candidate failure
Brian Springhthorpe

Symposium Grid -- Division of Chemical Toxicology -- Session Listing

Symposium Grid -- Drug Discovery -- Session Listing

The 232nd ACS National Meeting, San Francisco, CA, September 10-14, 2006