Hybrid polymers with reversible hydrophobic regions by combination of RAFT and ATRP

POLY 482

Krishnan Ranganathan, Rajesh K Kainthan, Donald E Brooks, don.brooks@ubc.ca, and Jayachandran N Kizhakkedathu. Department of Pathology and Laboratory Medicine, Chemistry and Centre for Blood Research, University of British Columbia, 2350 Health Sciences Mall, Life Sciences Centre, Vancouver, BC V6T 1Z3, Canada
Abstract: Double hydrophilic hybrid copolymers of PDMA/PNIPAm were synthesized by a combination of RAFT and ATRP “living” radical polymerizations from a multi functionalized hyperbranched polyglycerol (HPG) core. The incorporation of ATRP and azo initiator was achieved by the derivatization of hydroxyl groups (–OH) of the hyperbranched polyglycerol core. Azo initiator and S,S'-bis(a,a'-dimethyl-a''-acetic acid)trithiocarbonate CTA were utilized for RAFT polymerization of N,N-dimethylacrylamide. The polymerization of NIPAm from polyglycerol core was achieved by ATRP polymerization with HMTETA/Cu(I)Cl and Me6TREN/Cu(I)Cl catalysts at room temperature. Hybrid polymers with various molecular weights and narrow polydispersity were synthesized by adjusting the reaction conditions. The Me6TREN/Cu(I)Cl/(Cu(II)Cl2) catalyst system produced high molecular weights of PNIPAm than the HMTETA/Cu(I)Cl/Cu(II)Cl2 catalyst. At certain compositions of PDMA and PNIPAM, these hybrid polymers produced stable water soluble nanoaggregates above the LCST of PNIPAm (35 oC). With increase in the amount of PNIPAm, the hybrid polymers precipitated from aqueous solution above LCST. These hybrid polymers with reversible hydrophobic regions could be potential candidates for the delivery of hydrophobic drugs at physiological temperature
 

Nanoparticles and Microparticles: Synthesis and Applications
6:00 PM-8:00 PM, Tuesday, 12 September 2006 Moscone Center -- Hall D, Poster

Sci-Mix
8:00 PM-10:00 PM, Monday, 11 September 2006 Moscone Center -- Hall D, Sci-Mix

Division of Polymer Chemistry

The 232nd ACS National Meeting, San Francisco, CA, September 10-14, 2006