| MEDI | Sunday, 26 March 2006 | ||
8:30 AM-12:35 PM Georgia World Congress Center -- Georgia Ballroom 1, Oral | |||
11-Beta Hydroxysteroid Dehydrogenase | |||
| Organizer: | James M. Balkovec | ||
| 8:30 AM | Introductory Remarks | ||
| 8:35 AM | 1 | 11β-Hydroxysteroid dehydrogenase type 1 as a therapeutic target in metabolic syndrome and beyond Brian R Walker, Jonathan R Seckl | |
| 9:35 AM | 2 | Substituted adamantanamides as novel inhibitors of 11β-hydroxysteroid dehydrogenase type 1 Joannes TM Linders, Gustaaf HM Willemsens, Danny Bellens, Christophe Buyck, Peter De Backker, Kantharaj Ethirajulu, Ron AHJ Gilissen, Brian Hrupka, Libuse Jaroskova, Guy van Lommen, Ann Meulemans, Karine Smans, Pascal van Dorsselaer, Louis Van der Veken, Monique Berwaer | |
| 10:15 AM | 3 | Beta-keto sulfones and beta-keto sulfonamides as selective inhibitors of the 11beta-HSD1 Jason S. Xiang, Vipin Suri, Steve Tam, John C. McKew, Manus Ipek, Lihren Chen, Nelson Huang, Jianchang Li, Wei Li, Henry Lombart, Tarek Mansour, Jill Nunez, May Tam, Charlie Wu, Yuzhe Xin, Xin Xu, Yanling Zhang, James Tobin | |
| 10:45 AM | 4 | Structural insights into 11B-HSD1 function and inhibition David J Hosfield | |
| 11:25 AM | 5 | Bicyclo[2.2.2]octyltriazole inhibitors of 11ß-HSD1 Sherman T. Waddell, Xin Gu, Gina Santorelli, Donald Graham, James Balkovec | |
| 12:05 PM | 6 | 11beta-Hydroxysteroid dehydrogenase type 1 (11beta-HSD1) inhibition prolonged memory retention in mice Beatriz A. Rocha | |
Symposium Grid -- Division of Medicinal Chemistry -- Session Listing
Symposium Grid -- Drug Discovery -- Session Listing
The 231st ACS National Meeting, Atlanta, GA, March 26-30, 2006