| MEDI | Sunday, 28 August 2005 | ||
1:30 PM-5:30 PM Washington DC Convention Center -- Ballroom A, Oral | |||
Approaches to the Treatment of Anxiety and Depression | |||
| Sponsored by Teledyne Isco | |||
| Organizer, Presiding: | Andrew Stamford | ||
| 1:30 PM | Introductory Remarks | ||
| 2:10 PM | 16 | Identification and in vivo characterization of allosteric modulators of the GABAA ion channel with functional selectivity for the a3b3g2 subtype David J. Hallett, John R. Atack, J. Luis Castro, Susan Cook, Robert W. Carling, Rebecca Dias, Gerard R. Dawson, Simon Goodacre, Alexander Humphries, Sarah Kelly, Rachel J. Lincoln, George R. Marshall, Ruth M. McKernan, Leslie J. Street, David S. Reynolds, Michael G. N. Russell, Alison Smith, Wayne F. A. Sheppard, Joanne L. Stanley, Spencer Tye, Keith A. Wafford, Paul J. Whiting | |
| 2:50 PM | 17 | Discovery of a potent, selective and orally active 5-HT6 receptor agonist, WAY-181187 Derek C. Cole, Joseph R. Stock, William J. Lennox, Ronald C. Bernotas, John W. Ellingboe, Louis Leung, Deborah Smith, Gouming Zhang, Ping Li, Lin Qian, Lee A. Dawson, Steve Boikess, Sharon Rosenzweig-Lipson, Chad E. Beyer, Lee E. Schechter | |
| 3:30 PM | 18 | Design and synthesis of tricyclic corticotropin-releasing factor-1 (CRF1) antagonists John P Williams | |
| 4:10 PM | 19 | Design and synthesis of constrained imidazoles as CRF1R antagonists Xiaojun Han, Jodi Michne, Edward Ruediger, Rita Civiello, Sokhom Pin, Kevin Burris, Lynn Balanda, Lawrence Fung, Jay Knipe, Shelly Ren, Dedong Wu, Qi Gao, Stella Huang, Tracey Fiedler, Kaitlin Browman, Robert Macci, Matthew Taber, Jie Zhang, Gene Dubowchik | |
| 4:50 PM | 20 | Topology II CRF–1 receptor antagonists Raymond F Horvath, J Kehne, D Hoffman, R Brodbeck, L Fung, Y Yamaguchi | |
Symposium Grid -- Division of Medicinal Chemistry -- Session Listing
The 230th ACS National Meeting, in Washington, DC, Aug 28-Sept 1, 2005