MEDISunday, 28 August 2005

9:00 AM-12:20 PM Washington DC Convention Center -- 146A, Oral
General Oral Session
Organizer:David Rotella
Presiding:Jeff A. Zablocki
9:00 AMMultiple 5-HT approaches to novel anti-depressants
Simon E Ward
9:20 AMSynthesis and structure-activity relationship of tricyclic piperidinylidenes and tropanylidenes, a novel class of delta opioid agonists
Bart L. De Corte, John R Carson, Andrea B Works, Christine M Razler, Mark E. McDonnell, James J. McNally, Li Liu, Philip M. Pitis, Laura Andraka, Christopher A Teleha, Jef C. Proost, Sui-Po Zhang, Ellen E. Codd, Raymond W. Colburn, Dennis J. Stone, Lory J. Molino, Christopher R. Van Besien, Christopher M. Flores, Scott L. Dax
9:40 AMSynthesis of small molecules designed to complement disease-associated thyroid hormone receptor mutants
A. Quamrul Hassan, John T. Koh
10:00 AMCDK2/CyclinA inhibitors: Targeting the cyclinA recruitment site with small molecules derived from peptide leads
Daniel P. Sutherlin, Georgette M. Castanedo, Kevin Clark, Shumei Wang, Vickie Tsui, Mengling Wong, John B. Nicholas, Dineli Wickramasinghe, James Marsters
10:20 AMNovel VEGFR-2 kinase inhibitors for the treatment of cancer
Stephen J. Boyer, Jennifer M. Burke, Catherine R. Brennan, Warren Brini, William Collibee, Julie A. Dixon, Jacques Dumas, Frederick Ehrgott, Holia Hatoum-Mokdad, Zhenqui Hong, Harold C. Kluender, Wendy Lee, Xin Ma, Raymond Reeves, Robert N. Sibley, Tiffany Turner, Wai Wong, Yanlin Zhang, Cheryl Brink, Christopher Carter, Yong Chang, Du-Shieng Chien, Christian Cortes, James Elting, Randall M. Jones, Mark McHugh, Adrienne Natrillo, Barbara Polony, Patrick Vincent, Dean Wilkie, Deborah Webb, Guochang Zhu
10:40 AMSynthesis and characterization of 2,4-diaryl-2,5-dihydropyrrole inhibitors of the mitotic kinesin KSP: N1-Ureas and C2-phenols
Robert M. Garbaccio, Edward S. Tasber, Mark E. Fraley, George D. Hartman, Robert B. Lobell, Carolyn A. Buser, Weikang Tao, Hans E. Huber, Nancy E. Kohl, Lawrence C. Kuo, Youwei Yan, Maricel Torrent, Thomayant Prueksaritanont, Donald Slaughter
11:00 AMPolyaminohydroxamic acid derivatives as histone deacetylase (HDAC) inhibitors
Sheeba Varghese, Anchalee Jiemjit, Steven D. Gore, Tiffany Baran, Robert A. Casero, Patrick M. Woster
11:20 AMSupramolecular photonic therapeutic agents: pH Responsive anti-cancer drugs
Donal F. O'Shea, Shane McDonnell, Michael Hall
11:40 AMDesign and synthesis of an array of selective androgen receptor modulators
Ryan P. Trump, Philip Turnbull, Jean-Baptiste E. Blanc, Robert W. Wiethe, Eugene L. Stewart, Matilde Caivano, David Gray, William J. Hoekstra, Timothy M. Willson
12:00 PMNovel potent allosteric inhibitors of HCV NS5B polymerase
Christian Brochu, René Coulombe, J. R. Gillard, E. Jolicoeur, Peter Kohlbauer, Peter Kühn, Marc-André Poupart, Sylvain Lefebvre, Ginette McKercher, George Kukolj, P. L. Beaulieu

Symposium Grid -- Division of Medicinal Chemistry -- Session Listing

The 230th ACS National Meeting, in Washington, DC, Aug 28-Sept 1, 2005